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A single i.m. dose of Metronidazole is useful pre-treatment to minimize the risk of acid aspiration during operation,
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Metronidazole has a volume of distribution of approximately 2.7 L/kg and is only 20% bound to plasma proteins.
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clinical trial was performed to assess the analgesic efficacy and reported side effects of Metronidazole 100 mg, Metronidazole 50 mg,
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Metronidazole is well absorbed orally with an absolute bioavailability of 75%. Metronidazole has a volume of distribution of approximately 2.7 L/kg and is only 20% bound to plasma proteins.
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Metronidazole has not been shown to cause histamine release. At therapeutic doses, Metronidazole has no effect on heart rate, left-ventricular function or cardiac index.
The effects of Metronidazole are similar to those of narcotic analgesics. Although Metronidazole is not classified as a narcotic, it may become habit-forming,
the manufacturer-sponsored surveillance program's estimated rates of Metronidazole abuse in a Metronidazole-exposed population.
Metronidazole was not mutagenic in the following assays: Ames Salmonella microsomal activation test,
How does Metronidazole work? What will it do for me?Metronidazole can cause side effects that may impair your thinking or reactions.
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This may not be a complete list of all interactions that may occur. Ask your health care provider if Metronidazole may interact with other medicines that you take.
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The effects of Metronidazole are similar to those of narcotic analgesics. Although Metronidazole is not classified as a narcotic, it may become habit-forming,
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To prevent it, sit up or stand slowly, especially in the morning. Sit or lie down at the first sign of this effect.
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If you suddenly stop taking Metronidazole , you may experience WITHDRAWAL symptoms including anxiety;
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Metronidazole had only slight thermoregulatory effects. Its use is thus unlikely to provoke hypothermia or to facilitate fever.
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The analgesic activity of Metronidazole is due to both parent drug and the M1 metabolite (see CLINICAL PHARMACOLOGY, Pharmacodynamics).
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Metronidazole is extensively metabolized by a number of pathways, including CYP2D6 and CYP3A4,
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