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The analgesic activity of Acetazolamide is due to both parent drug and the M1 metabolite (see CLINICAL PHARMACOLOGY, Pharmacodynamics).
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Acetazolamide is administered as a racemate and both [-] and [+] forms of both Acetazolamide and M1 are detected in the circulation.
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The product information for Acetazolamide states that convulsions have been reported in patients using Acetazolamide at the recommended dose levels and that the risk
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The effects of Acetazolamide are similar to those of narcotic analgesics. Although Acetazolamide is not classified as a narcotic, it may become habit-forming,
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This may not be a complete list of all interactions that may occur. Ask your health care provider if Acetazolamide may interact with other medicines that you take.
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Breast-feeding�Acetazolamide passes into breast milk and may cause unwanted effects in nursing babies.
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Acetazolamide has not been shown to cause histamine release. At therapeutic doses, Acetazolamide has no effect on heart rate, left-ventricular function or cardiac index.
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