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Talk with your doctor if Prometrium stops working well. Do not take more than prescribed.Some people who use Prometrium for a long time without a break may develop a physical need to continue taking it.
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Do not stop using this medication suddenly without first talking to your doctor.
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In general, both enantiomers of Prometrium and M1 follow a parallel time course in the body following single and multiple doses although small differences (~10%) exist in the absolute amount of each enantiomer present.
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Prometrium and M1 elimination half-lives (13 hrs. for Prometrium and 19 hrs. for M1).
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Prometrium is well absorbed orally with an absolute bioavailability of 75%. Prometrium has a volume of distribution of approximately 2.7 L/kg and is only 20% bound to plasma proteins.
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This is known as physical DEPENDENCE. If you suddenly stop taking Prometrium , you may experience WITHDRAWAL symptoms including anxiety;
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which may affect the therapeutic response (see PRECAUTIONS - Drug Interactions).
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Prometrium may not work as well and may require higher doses to obtain the same effect as when originally taken.
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Tell your doctor or dentist that you take Prometrium before you receive any medical or dental care, emergency care, or surgery.
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Linear pharmacokinetics have been observed following multiple doses of 50 and 100 mg to steady-state.Racemic Prometrium is rapidly and almost completely absorbed after oral administration.
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