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Metronidazole is found in breast milk. Do not breast-feed while taking Metronidazole .When used for long periods of time or at high doses,
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Metronidazole should be used during pregnancy only if the potential benefit justifies the potential risk to the fetus.
Metronidazole was evaluated in peri- and post-natal studies in rats.
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Metronidazole was not mutagenic in the following assays:
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No effects on fertility were observed for Metronidazole at oral dose levels up to 50 mg/kg,
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Metronidazole was not mutagenic in the following assays: Ames Salmonella microsomal activation test,
more potent than Metronidazole in producing analgesia and 200 times more potent in ?-opioid binding.
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Metronidazole may rarely be habit forming. Metronidazole should be avoided in patients with a history of opiate addiction or hypersensitivity to opiate medications.
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The binding of Metronidazole to human plasma proteins is approximately 20%,
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Linear pharmacokinetics have been observed following multiple doses of 50 and 100 mg to steady-state.Racemic Metronidazole is rapidly and almost completely absorbed after oral administration.
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The volume of distribution of Metronidazole was 2.6 and 2.9 liters/kg in male and female subjects, respectively,
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Taking more than the prescribed amount of this medication could result in seizures or decreased breathing.
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