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    Diltiazem has not been shown to cause histamine release. At therapeutic doses, Diltiazem has no effect on heart rate, left-ventricular function or cardiac index.
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    Diltiazem is extensively metabolized by a number of pathways, including CYP2D6 and CYP3A4, as well as by conjugation of parent and metabolites.
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    Linear pharmacokinetics have been observed following multiple doses of 50 and 100 mg to steady-state.Racemic Diltiazem is rapidly and almost completely absorbed after oral administration.
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