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Metronidazole should be used during pregnancy only if the potential benefit justifies the potential risk to the fetus.
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Although Metronidazole is known to exhibit a local anaesthetic effect, how Metronidazole exerts this effect is not understood fully.
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since observed maximal placoncentrations after multiple oral doses are higher than expected based on single-dose data.
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Metronidazole is administered as a racemate and both [-] and [+] forms of both Metronidazole and M1 are detected in the circulation.
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Metronidazole is well absorbed orally with an absolute bioavailability of 75%. Metronidazole has a volume of distribution of approximately 2.7 L/kg and is only 20% bound to plasma proteins.
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1 Dosing may be increased to 100 mg every four to six hours, but the daily dosage should not exceed 400 mg 1 and should be limited to 250 to 300 mg .
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This indicates that Metronidazole slightly decreases the precision of thermoregulatory control in addition to reducing the setpoint.
The binding of Metronidazole to human plasma proteins is approximately 20%,
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Metronidazole had only slight thermoregulatory effects. Its use is thus unlikely to provoke hypothermia or to facilitate fever.
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Use Metronidazole with caution in the ELDERLY; they may be more sensitive to its effects.Metronidazole should not be used in CHILDREN younger than 16 years old;
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In an open randomized trial, rectal Metronidazole was compared with our standard treatment acetaminophen/codeine suppositories. We expected Metronidazole to be equally effective as our current standard but with fewer side effects.
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