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Linear pharmacokinetics have been observed following multiple doses of 50 and 100 mg to steady-state.Racemic Moduretic is rapidly and almost completely absorbed after oral administration.
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Moduretic has been shown to inhibit reuptake of norepinephrine and serotonin in vitro,
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This indicates that Moduretic slightly decreases the precision of thermoregulatory control in addition to reducing the setpoint.
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Moduretic may rarely be habit forming. Moduretic should be avoided in patients with a history of opiate addiction or hypersensitivity to opiate medications.
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To prevent it, sit up or stand slowly, especially in the morning. Sit or lie down at the first sign of this effect.
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