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The mean absolute bioavailability of a 100 mg oral dose is approximately 75%. The mean peak plasma concentration of racemic Motilium and M1 occurs at two and three hours, respectively, after administration in healthy adults.
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In general, both enantiomers of Motilium and M1 follow a parallel time course in the body following single and multiple doses although small differences (~10%) exist in the absolute amount of each enantiomer present.
The effects of Motilium and its metabolite mono-O-demethyl-Motilium,
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clinical trial was performed to assess the analgesic efficacy and reported side effects of Motilium 100 mg, Motilium 50 mg,
The analgesic activity of Motilium is due to both parent drug and the M1 metabolite (see CLINICAL PHARMACOLOGY, Pharmacodynamics).
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