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Acetazolamide was evaluated in peri- and post-natal studies in rats.
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Acetazolamide is well absorbed orally with an absolute bioavailability of 75%. Acetazolamide has a volume of distribution of approximately 2.7 L/kg and is only 20% bound to plasma proteins.
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Linear pharmacokinetics have been observed following multiple doses of 50 and 100 mg to steady-state.Racemic Acetazolamide is rapidly and almost completely absorbed after oral administration.
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Check the label on the medicine for exact dosing instructions.Acetazolamide may cause drowsiness and dizziness.
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