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adjustment of the dosing regimen is recommended (see DOSAGE AND ADMINISTRATION).
1 Dosing may be increased to 100 mg every four to six hours, but the daily dosage should not exceed 400 mg 1 and should be limited to 250 to 300 mg .
Although Tacrolimus is known to exhibit a local anaesthetic effect, how Tacrolimus exerts this effect is not understood fully.
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In general, both enantiomers of Tacrolimus and M1 follow a parallel time course in the body following single and multiple doses although small differences (~10%) exist in the absolute amount of each enantiomer present.
We expected Tacrolimus to be equally effective as our current standard.
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The binding of Tacrolimus to human plasma proteins is approximately 20%,
tests indicates that Tacrolimus does not pose a genotoxic risk to humans.
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Tacrolimus can impair thinking and the physical abilities required for driving or operating machinery. Tacrolimus should be avoided in patients intoxicated with alcohol,
Tacrolimus has both opioid and monoaminergic agonist actions.
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