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Acetazolamide may induce psychic and physical dependence of the morphine-type (?- opioid) (See WARNINGS).
To prevent it, sit up or stand slowly, especially in the morning. Sit or lie down at the first sign of this effect.
Acetazolamide has not been shown to cause histamine release. At therapeutic doses, Acetazolamide has no effect on heart rate, left-ventricular function or cardiac index.
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Use Acetazolamide with caution in the ELDERLY; they may be more sensitive to its effects.Acetazolamide should not be used in CHILDREN younger than 16 years old;
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Nalbuphine consumption in the first 24 h after operation was reduced by 35% in the Acetazolamide group.
which may affect the therapeutic response (see PRECAUTIONS - Drug Interactions). Acetazolamide and its metabolites are excreted primarily in he urine with observed plasma half-lives of 6.3 and 7.4 hours for Acetazolamide and M1, respectively.
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since observed maximal placoncentrations after multiple oral doses are higher than expected based on single-dose data.
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