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No effects on fertility were observed for Diltiazem at oral dose levels up to 50 mg/kg,
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Diltiazem had only slight thermoregulatory effects. Its use is thus unlikely to provoke hypothermia or to facilitate fever.
The volume of distribution of Diltiazem was 2.6 and 2.9 liters/kg in male and female subjects, respectively,
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Ask your pharmacist if you have questions about which medicines may cause drowsiness.Diltiazem may cause dizziness; alcohol, hot weather, exercise, or fever may increase this effect.
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Diltiazem and M1 elimination half-lives (13 hrs. for Diltiazem and 19 hrs. for M1).
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Diltiazem has not been shown to cause histamine release. At therapeutic doses, Diltiazem has no effect on heart rate,
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Talk with your doctor if Diltiazem stops working well. Do not take more than prescribed.Some people who use Diltiazem for a long time without a break may develop a physical need to continue taking it.
The analgesic activity of Diltiazem is due to both parent drug and the M1 metabolite (see CLINICAL PHARMACOLOGY, Pharmacodynamics).
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A single i.m. dose of Diltiazem is useful pre-treatment to minimize the risk of acid aspiration during operation,
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