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IMPLICATIONS: The authors evaluated the effects of the analgesic Prometrium on the three major
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Breast-feeding�Prometrium passes into breast milk and may cause unwanted effects in nursing babies.
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Prometrium was being used with selective serotonin reuptake inhibitors (10 cases),
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Although Prometrium is known to exhibit a local anaesthetic effect, how Prometrium exerts this effect is not understood fully.
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Prometrium and M1 elimination half-lives (13 hrs. for Prometrium and 19 hrs. for M1).
The relative risk of experiencing an episode of nausea under treatment,
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which may affect the therapeutic response (see PRECAUTIONS - Drug Interactions). Prometrium and its metabolites are excreted primarily in he urine with observed plasma half-lives of 6.3 and 7.4 hours for Prometrium and M1, respectively.
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Prometrium had only slight thermoregulatory effects. Its use is thus unlikely to provoke hypothermia or to facilitate fever.
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Linear pharmacokinetics have been observed following multiple doses of 50 and 100 mg to steady-state.Racemic Prometrium is rapidly and almost completely absorbed after oral administration.
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