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Linear pharmacokinetics have been observed following multiple doses of 50 and 100 mg to steady-state.Racemic Ropinirole is rapidly and almost completely absorbed after oral administration.
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Ropinirole has a volume of distribution of approximately 2.7 L/kg and is only 20% bound to plasma proteins.
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which may affect the therapeutic response (see PRECAUTIONS - Drug Interactions). Ropinirole and its metabolites are excreted primarily in he urine with observed plasma half-lives of 6.3 and 7.4 hours for Ropinirole and M1, respectively.
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Ropinirole 100 mg was statistically superior to placebo for TOTPAR, SPID, and time of remedication,
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Ropinirole has not been shown to cause histamine release. At therapeutic doses, Ropinirole has no effect on heart rate,
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Ropinirole is administered as a racemate and both [-] and [+] forms of both Ropinirole and M1 are detected in the circulation.
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